About: Funapide

An Entity of Type: book, from Named Graph: http://dbpedia.org, within Data Space: dbpedia.org

Funapide (INN) (former developmental code names TV-45070 and XEN402) is a novel analgesic under development by (formerly in partnership with Teva Pharmaceutical Industries) for the treatment of a variety of chronic pain conditions, including osteoarthritis, neuropathic pain, postherpetic neuralgia, and erythromelalgia, as well as dental pain. It acts as a small-molecule Nav1.7 and Nav1.8 voltage-gated sodium channel blocker. Funapide is being evaluated in humans in both oral and topical formulations, and as of July 2014, has reached phase IIb clinical trials.

Property	Value
dbo:abstract	Funapide (INN) (former developmental code names TV-45070 and XEN402) is a novel analgesic under development by (formerly in partnership with Teva Pharmaceutical Industries) for the treatment of a variety of chronic pain conditions, including osteoarthritis, neuropathic pain, postherpetic neuralgia, and erythromelalgia, as well as dental pain. It acts as a small-molecule Nav1.7 and Nav1.8 voltage-gated sodium channel blocker. Funapide is being evaluated in humans in both oral and topical formulations, and as of July 2014, has reached phase IIb clinical trials. (en)
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dbp:routesOfAdministration	dbr:Oral_administration dbr:Topical_medication
dbp:smiles	C1C2C5=CC6=COCO6 (en)
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rdfs:comment	Funapide (INN) (former developmental code names TV-45070 and XEN402) is a novel analgesic under development by (formerly in partnership with Teva Pharmaceutical Industries) for the treatment of a variety of chronic pain conditions, including osteoarthritis, neuropathic pain, postherpetic neuralgia, and erythromelalgia, as well as dental pain. It acts as a small-molecule Nav1.7 and Nav1.8 voltage-gated sodium channel blocker. Funapide is being evaluated in humans in both oral and topical formulations, and as of July 2014, has reached phase IIb clinical trials. (en)
rdfs:label	Funapide (en)
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