About: Mebolazine

An Entity of Type: chemical substance, from Named Graph: http://dbpedia.org, within Data Space: dbpedia.org

Mebolazine (INN; brand names Dostalon and Roxilon; also known as dimethazine, dymethazine, di(methasterone) azine, or 2α,17α-dimethyl-5α-androstan-17β-ol-3-one azine) is a synthetic, orally active androgen/anabolic steroid (AAS) and a 17α-alkylated derivative of dihydrotestosterone (DHT) which is no longer marketed. It has a unique and unusual chemical structure, being a dimer of methasterone linked at the 3-position of the A-ring by an azine group, and reportedly acts as a prodrug of methasterone.

Property	Value
dbo:abstract	Mebolazine (INN; brand names Dostalon and Roxilon; also known as dimethazine, dymethazine, di(methasterone) azine, or 2α,17α-dimethyl-5α-androstan-17β-ol-3-one azine) is a synthetic, orally active androgen/anabolic steroid (AAS) and a 17α-alkylated derivative of dihydrotestosterone (DHT) which is no longer marketed. It has a unique and unusual chemical structure, being a dimer of methasterone linked at the 3-position of the A-ring by an azine group, and reportedly acts as a prodrug of methasterone. Since 2008, mebolazine has been used illegally as an ingredient is some dietary supplements, including vitamin B supplements, and in the United States the Food and Drug Administration has taken legal action against such manufacturers. (en)
dbo:alternativeName	Dostalon, Roxilon (en)
dbo:casNumber	3625-07-8
dbo:fdaUniiCode	69C642I19V
dbo:pubchem	9571069
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dbp:casNumber	3625-07-08 (xsd:date)
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dbp:image	Mebolazine molecule ball.png (en)
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dbp:pubchem	9571069 (xsd:integer)
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dbp:stdinchikey	POPWFGNRCCUJGU-QQZDHCPGSA-N (en)
dbp:synonyms	Dimethazine; Dymethazine; Dimethasterone azine; Di azine; 2α,17α-Dimethyl-5α-androstan-17β-ol-3-one azine (en)
dbp:tradename	Dostalon, Roxilon (en)
dbp:unii	69 (xsd:integer)
dbp:verifiedfields	changed (en)
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gold:hypernym	dbr:Steroid
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rdfs:comment	Mebolazine (INN; brand names Dostalon and Roxilon; also known as dimethazine, dymethazine, di(methasterone) azine, or 2α,17α-dimethyl-5α-androstan-17β-ol-3-one azine) is a synthetic, orally active androgen/anabolic steroid (AAS) and a 17α-alkylated derivative of dihydrotestosterone (DHT) which is no longer marketed. It has a unique and unusual chemical structure, being a dimer of methasterone linked at the 3-position of the A-ring by an azine group, and reportedly acts as a prodrug of methasterone. (en)
rdfs:label	Mebolazine (en)
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