Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonist and also glycine receptor antagonist with similar potency and nicotinic acetylcholine receptors to a much lesser extent. It has powerful convulsant activity and should not be used in seizure-prone individuals.

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dbo:abstract
  • Il tiocolchicoside è una molecola solforata semisintetica derivata dal colchicoside, un glucoside prodotto dal colchico. Ha effetto miorilassante e viene utilizzato per il trattamento delle contratture muscolari.
  • Le thiocolchicoside est un dérivé semi-synthétique de la colchicine, il est utilisé comme médicament myorelaxant (noms commerciaux Coltramyl, Miorel)
  • Tiocolchicósido é um fármaco utilizado pela medicina como miorrelaxante.
  • Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonist and also glycine receptor antagonist with similar potency and nicotinic acetylcholine receptors to a much lesser extent. It has powerful convulsant activity and should not be used in seizure-prone individuals.
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  • 602-41-5
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  • T1X8S697GT
dbo:iupacName
  • N-[(7S)-3-(β-(D)-Glucopyranosyloxy)-1,2-dimethoxy-10-(methylsulfanyl)-9-oxo-5,6,7,9-tetrahydrobenzo[a]heptalen-7-yl]acetamide
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  • N-[-3--1,2-dimethoxy-10--9-oxo-5,6,7,9-tetrahydrobenzo[a]heptalen-7-yl]acetamide
dbp:kegg
  • D07276
dbp:legalStatus
  • Rx-only
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rdfs:comment
  • Il tiocolchicoside è una molecola solforata semisintetica derivata dal colchicoside, un glucoside prodotto dal colchico. Ha effetto miorilassante e viene utilizzato per il trattamento delle contratture muscolari.
  • Le thiocolchicoside est un dérivé semi-synthétique de la colchicine, il est utilisé comme médicament myorelaxant (noms commerciaux Coltramyl, Miorel)
  • Tiocolchicósido é um fármaco utilizado pela medicina como miorrelaxante.
  • Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonist and also glycine receptor antagonist with similar potency and nicotinic acetylcholine receptors to a much lesser extent. It has powerful convulsant activity and should not be used in seizure-prone individuals.
rdfs:label
  • Thiocolchicoside
  • Tiocolchicoside
  • Tiocolchicósido
  • Thiocolchicoside
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