Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonist and also glycine receptor antagonist with similar potency and nicotinic acetylcholine receptors to a much lesser extent. It has powerful convulsant activity and should not be used in seizure-prone individuals. This mechanism of action would be expected to induce withdrawal symptoms in gabaminergic (ex.
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- Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonist and also glycine receptor antagonist with similar potency and nicotinic acetylcholine receptors to a much lesser extent. It has powerful convulsant activity and should not be used in seizure-prone individuals. This mechanism of action would be expected to induce withdrawal symptoms in gabaminergic (ex. benzodiazepines, barbiturates, carbamates, ethanol) dependent individuals, including the potentially lethal delerium tremens.
- Le thiocolchicoside est un dérivé semi-synthétique de la colchicine, il est utilisé comme médicament myorelaxant (noms commerciaux Coltramyl, Miorel)
- Il tiocolchicoside è una molecola solforata semisintetica derivata dal colchicoside, un glucoside prodotto dal colchico. Ha effetto miorilassante e viene utilizzato per il trattamento delle contusioni muscolari.
- Tiocolchicósido é um fármaco utilizado pela medicina como miorrelaxante.
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- N-[(7S)-3-(β-(D)-Glucopyranosyloxy)-1,2-dimethoxy-10-(methylsulfanyl)-9-oxo-5,6,7,9-tetrahydrobenzo[a]heptalen-7-yl]acetamide
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- N-[-3--1,2-dimethoxy-10--9-oxo-5,6,7,9-tetrahydrobenzo[a]heptalen-7-yl]acetamide
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- LEQAKWQJCITZNK-MSQQGMGVSA-N
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- Le thiocolchicoside est un dérivé semi-synthétique de la colchicine, il est utilisé comme médicament myorelaxant (noms commerciaux Coltramyl, Miorel)
- Il tiocolchicoside è una molecola solforata semisintetica derivata dal colchicoside, un glucoside prodotto dal colchico. Ha effetto miorilassante e viene utilizzato per il trattamento delle contusioni muscolari.
- Tiocolchicósido é um fármaco utilizado pela medicina como miorrelaxante.
- Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonist and also glycine receptor antagonist with similar potency and nicotinic acetylcholine receptors to a much lesser extent. It has powerful convulsant activity and should not be used in seizure-prone individuals. This mechanism of action would be expected to induce withdrawal symptoms in gabaminergic (ex.
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- Thiocolchicoside
- Tiocolchicoside
- Thiocolchicoside
- Tiocolchicósido
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